Tuesday, January 29, 2013

GRANULES

GRANULES



Granules are aggregations of fine particles of powders in a mass of about spherical shape. They typically fall within the range of 850 µm to 4.75 mm size. They are particularly suitable for the preparation of solutions or mixtures of drugs, such as antibiotics, that are unstable in the presence of water.






Types of Granules

1.      Sustained release granules
These granules are intended to be used to achieve long term action of medicament.These are prepared on the bases of delayed time release technology.
Example of sustained release is Zmax SR containing azithromycine sustained release granules.
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2.      Enteric coated granules.
These are made to have action in intestine by preventing dissolution in stomach.Example  Abprazole™ sachets of enteric coated blue colored granules containing Omeprazole 25%w/w for equine use for both the treatment and prevention of Equine Gastric Ulcers (EGUS)
3.      Effervescent granules.
      Effervescent granules contain sodium bicarbonate and citric acid or tartaric acid in addition to the active ingredients. On solution in water, carbon dioxide is released. These forms mask the unpleasant taste anensure better absorption of the medications.



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